Sacubitril
Entresto is the only sacubitril product listed here, pairing 24 mg sacubitril with 26 mg valsartan in a single tablet to treat Heart Failure.
Key points
- The combination lowers the risk of death and hospitalization in adults with certain types of heart failure, used alongside other medications.
- Do not take Entresto during pregnancy: the combination may cause death or serious injury to the fetus in the last six months.
- Entresto is also used to treat certain types of heart failure in children aged 1 year and older.
How does sacubitril work?
Sacubitril blocks an enzyme called neprilysin, which breaks down signalling molecules that regulate blood volume and vessel width. With neprilysin inhibited, those molecules stay active longer, easing the workload on a heart that cannot pump efficiently. Valsartan adds a second action: it blocks a natural substance that tightens blood vessels, so blood flows more smoothly. The two ingredients work in parallel to reduce the strain a failing heart carries.
